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產(chǎn)品基本信息
產(chǎn)品編號:G797425
產(chǎn)品名稱:Uprosertib
產(chǎn)品CAS:1047634-65-0
規(guī)格含量:5mg
產(chǎn)品價格:面議
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產(chǎn)品詳細介紹
標準品編號:
G797425
名稱:
Uprosertib
別名:
N-[(1S)-2-Amino-1-[(3,4-difluorophenyl)methyl]ethyl]-5-chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)-2-furancarboxamide; GSK 2141795C
CAS號:
1047634-65-0
分子式:
C??H??Cl?F?N?O?
分子量:
429.25
種類:
Standards; Enzyme Activators and Inhibitors;
應(yīng)用:
Uprosertib is a potent and selective inhibitor of pan-Akt (1). Serine/threonine protein kinases, such as Akt, play important roles in cellular activities including cell survival and apoptosis.
參考文獻
Seefield, M. A., et al.: PCT Int. Appl.(2008),WO2008098104A120080814; Liu, W., et al.: Toxicol. Appl. Pharmacol, 381, 114729 (2019);