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產(chǎn)品基本信息
產(chǎn)品編號(hào):L486320
產(chǎn)品名稱:LY2157299
產(chǎn)品CAS:700874-72-2
規(guī)格含量:10mg
產(chǎn)品價(jià)格:面議
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產(chǎn)品詳細(xì)介紹
標(biāo)準(zhǔn)品編號(hào):
L486320
名稱:
LY2157299
別名:
Galunisertib; 4-(2-(6-Methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinoline-6-carboxamide; 4-[5,6-Dihydro-2-(6-methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-6-quinolinecarboxamide
CAS號(hào):
700874-72-2
分子式:
C??H??N?O
外觀:
白色至白色固體
熔點(diǎn):
241-242°C
分子量:
369.42
儲(chǔ)存:
-20°C Freezer
溶解度:
DMSO (Slightly), Methanol (Slightly)
種類:
Research Tools; Enzyme Activators and Inhibitors;
應(yīng)用:
LY2157299 is a TGF-β type I receptor kinase inhibitor. LY2157299 has been used to inhance chemotherapy action against triple negative breast cancer (TNBC).
參考文獻(xiàn)
Bhola, N.E., et. al.: J. Clin. Invest., 123, 1348 (2013)