產(chǎn)品基本信息
產(chǎn)品編號(hào):Z150700
產(chǎn)品名稱:Zatebradine Hydrochloride
產(chǎn)品CAS:91940-87-3
規(guī)格含量:5mg
產(chǎn)品價(jià)格:面議
聯(lián)系我們:
產(chǎn)品詳細(xì)介紹
標(biāo)準(zhǔn)品編號(hào):
Z150700
名稱:
Zatebradine Hydrochloride
別名:
UL-FS 49; ULFS 49CL; 3-[3-[[2-(3,4-Dimethoxyphenyl)ethyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one Hydrochloride;
CAS號(hào):
91940-87-3
參考CAS號(hào):
Free Base: 85175-67-3
分子式:
C??H??N?O?•HCl
分子量:
456.573646
類別:
Standards; Enzyme Activators and Inhibitors;
應(yīng)用:
Zatebradine Hydrochloride exhibits bradycardic properties and blocks the hyperpolarization-activated cyclic nucleotide-gated (HCN). It is also a sinus node inhibitor.
參考文獻(xiàn)
Stieber, J., et al.: Mol. Pharmacol 69, 1328 (2006); Thollon, C., et al.:ÂBr. J. Pharmacol. 112, 37 (1992); Reiffen, M., et al.: J. Med. Chem. 33, 1496 (1990);ÂL Sen et al. J. Cardiovasc. Pharmacol. 7, 29Â(2007);