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產(chǎn)品基本信息
產(chǎn)品編號(hào):B377008
產(chǎn)品名稱:BIBU 1361 Dihydrochloride
產(chǎn)品CAS:1643609-75-9
規(guī)格含量:2.5mg
產(chǎn)品價(jià)格:面議
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產(chǎn)品詳細(xì)介紹
標(biāo)準(zhǔn)品編號(hào):
B377008
名稱:
BIBU 1361 Dihydrochloride
別名:
N-(3-Chloro-4-fluorophenyl)-6-[4-[(diethylamino)methyl]-1-piperidinyl]-pyrimido[5,4-d]pyrimidin-4-amine Dihydrochloride
CAS號(hào):
1643609-75-9
備用CAS:
Free Base: 793726-84-8
分子式:
C??H??ClFN? • 2(HCl)
外觀:
Yellow Solid
分子量:
443.9523646
儲(chǔ)存:
冰箱保存
溶解度:
DMSO (Slightly), Methanol (Very Slightly)
類別:
Standards; Enzyme Activators and Inhibitors;
應(yīng)用:
BIBU 1361 Dihydrochloride, is a potent inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase (IC50 = 3 nM). It also blocks downstream EGFR signaling events such as MAPKK/MAPK activation.
文獻(xiàn)
Download MSDS File